Degarelix acetate yog ib qho hluavtaws gonadotropin-tso cov tshuaj hormones (GnRH) receptor antagonist uas txo cov kev tso tawm ntawm gonadotropins thiab testosterone los ntawm reversibly khi rau GnRH receptor ntawm lub caj pas pituitary, yog li exerting anti-prostate cancer nyhuv.
Specifications
- Tshuaj Lub Npe: Acetyl-(2S)-N-[(2S,3S)-3-{[(2S)-1-[(2R)-2-hydroxy-3-(naphthalen -2-yl)propanoyl]pyrrolidine-2-carbonyl]amino}-2-{3-[4-(2-hydroxyethyl)-1-piperazinyl ]propyl}-3-methyl-L-valinamide
- Molecular Formula: C82H103ClN12O16
Molecular Luj: 1632.44 g / mol
- CAS Nr .: 214766-78-6
- Purity Ntau dua lossis sib npaug li 98 feem pua
- Impurity Tsawg dua lossis sib npaug rau 0.5 feem pua
- Pom: Dawb mus rau dawb hmoov
- Solubility: Soluble hauv dej thiab methanol
Daim ntawv thov
- Kev kho mob qog noj ntshav siab tshaj plaws: DEGARELIX yog gonadotropin-tso hormone (GnRH) receptor antagonist siv los txo cov theem ntawm testosterone hauv cov ntshav los kho mob qog noj ntshav prostate.
Vim li cas thiaj siv Degarelix Acetate:
Degarelix acetate yog cov tshuaj siv los kho mob qog noj ntshav prostate siab heev los ntawm kev thaiv cov tshuaj hormones uas txhawb kev loj hlob thiab kis ntawm cov qog nqaij hlav cancer. Nws yog gonadotropin-tso cov tshuaj hormones (GnRH) antagonist uas feem ntau siv thaum lwm txoj kev kho tshuaj hormone ua tsis tau lossis tsis ua haujlwm. Degarelix ua haujlwm sai kom txo qis testosterone qib thiab tuaj yeem ua rau txo qis hauv prostate loj thiab ua haujlwm qog noj ntshav. Nws yog siv raws li kev txhaj tshuaj subcutaneous thiab feem ntau zoo zam nrog qee qhov kev mob tshwm sim. Zuag qhia tag nrho, degarelix acetate yog ib qho kev kho mob tseem ceeb rau cov txiv neej uas mob qog noj ntshav siab.
Cia
- Khaws ntawm chav tsev kub ntawm 20-25 degree (68-77 degree F).
- Tiv thaiv los ntawm lub teeb thiab noo noo.
- Khaws kom deb ntawm cov menyuam yaus.
Cim npe nrov: Degarelix, Tuam Tshoj degarelix manufacturers, hoobkas











