Vildagliptin yog ib yam tshuaj uas muaj nyob rau hauv chav kawm ntawm dipeptidyl peptidase -4 inhibitors (DPP4) thiab feem ntau yog tshuaj los tswj cov ntshav qab zib hauv cov neeg mob ntshav qab zib hom 2. Nws ua haujlwm los ntawm inhibiting cov enzyme DPP4, uas ua rau nce insulin secretion thiab txo cov piam thaj hauv lub siab.
Specifications
Melting point: 153-155 degree
Kev sib hloov tshwj xeeb: -78.3 degree (c=9.73inmethanol)
Kub taw tes: 531.3 ± 5 0.0 degree (Predicted)
Qhov ceev: 1.27
Flash point: 275.1 degree
Solubility: Solublein DMSO (upto 45mg / ml), inDMF (upto 20mg / ml), orinEthanol (upto 20mg / ml).
Acidity coefficient: (pKa) 15.
Daim ntawv: khov
Xim: Dawb
Daim ntawv thov
Vildagliptin feem ntau yog qhia rau kev kho mob ntawm hom 2 mob ntshav qab zib mellitus. Nws yog feem ntau raug sau nrog kev noj zaub mov thiab kev tawm dag zog thiab siv tau ib leeg lossis ua ke nrog lwm cov tshuaj tiv thaiv kab mob ntshav qab zib (xws li metformin) txhawm rau txhim kho glycemic tswj. Cov tshuaj tsis yog npaj rau kev kho mob ntshav qab zib hom 1 lossis ntshav qab zib ketoacidosis.
Vim li cas thiaj siv Vildagliptine?
Vildagliptin yog ib qho kev xaiv, kev sib tw thiab thim rov qab DPP24 inhibitor. Glucose-dependent insulinotropic polypeptide (GIP) thiab glucagon-zoo li polypeptide 21 (GLP21) yog cov tshuaj hormones tseem ceeb rau kev tswj cov piam thaj hauv lub cev, thiab ob qho tib si muaj cov nyhuv incretin-stimulating.
Cia
Vildagliptin yuav tsum tau muab cia rau hauv chav tsev kub, kom deb ntawm tshav ntuj ncaj qha, noo noo, thiab cua sov. Cov tshuaj yuav tsum tau khaws cia rau hauv nws lub thawv qub, thiab lub thawv yuav tsum kaw kom zoo thaum tsis siv.
Cim npe nrov: Tuam Tshoj vildagliptin manufacturers, hoobkas











